Design, Synthesis and Fungicidal Activity of Triamide Compounds
Tolfenpyrad, a commercialized Pyrazolecarboxamide Derivatives, shows good insecticidal/acaricidal activity against Lepidoptera, Hemiptera, Thysanoptera and eriophyid mites in vegetables, ornamentals and fruit, also active against the fungus Sphaerotheca fuliginea. Chlorantraniliprole, discovered by Du pont, is a broad-spectrum insecticide with novel structure and new mechanism only acting on RyR distributed in insects. In this paper, using methods of active substructure combination and the intermediate derivatization method, a series of triamide compounds combining some structures of Tolfenpyrad and Chlorantraniliprole were designed, synthesized and bioassayed. The structure-activity relationships of the synthesized compounds were also discussed comprehensively.
triamide compounds active substructure combination intermediate derivatization method design and synthesis fungicidal activity
Lizeng Wang Changling Liu Xufeng Sun Zhinian Li Jie Lan Lanhui Ren Qiao Wu Huiwei Chi
State Key Laboratory of the Discovery and Development of Novel Pesticide, Shenyang Research Institute of Chemical Industry Co. Ltd. , Shenyang, China
国际会议
北京
英文
307
2012-09-15（万方平台首次上网日期，不代表论文的发表时间）